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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10299 | AMG PERK 44 | ERK | |
AMG PERK 44 is an orally active and selective PERK inhibitor (IC50: 6 nM) and induces autophagy. It has 1000-fold and 160-fold selectivity over GCN2 (IC50: 7300 nM) and B-Raf (IC50 >1000 nM), respectively. |